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Meperidine and Promethazine Capsules e Distúrbios convulsivos

Resultado da verificação da interação do medicamento Meperidine and Promethazine Capsules com doença Distúrbios convulsivos quanto a segurança no uso em conjunto.

Resultado da verificação:
Meperidine and Promethazine Capsules <> Distúrbios convulsivos
Relevância: 23.07.2019 Revisor: Shkutko P.M., M.D., in

Na verificação da interação, conforme informações das fontes confiáveis como Drugs.com, Rxlist.com, Webmd.com, Medscape.com, foram identificadas as contra-indicações ou efeitos colaterais que podem prejudicar a saúde ou aumentar efeito negativo ao consumir o medicamento com esta doença concomitante.

Consumidor:

Narcóticos opiáceos analgésicos, agentes podem exacerbar convulsões em pacientes com transtornos convulsivos e, em doses mais elevadas, têm sido relatados para induzir convulsões em pacientes sem história prévia de convulsões. O proconvulsant atividade pode ser maior com a meperidina, o metabólito ativo do que é pensado para ser responsável. A terapia com opióides devem ser administrados com precaução em doentes com predisposição para convulsões.

Referências
  • Strong WE, Matson M "Probable seizure after alfentanil." Anesth Analg 68 (1989): 692-3
  • Armstrong PJ, Bersten A "Normeperidine toxicity." Anesth Analg 65 (1986): 536-8
  • "Product Information. Dalgan (dezocine)." Astra USA, Westborough, MA.
  • "Product Information. Darvon (propoxyphene)." Lilly, Eli and Company, Indianapolis, IN.
  • Sebel PS, Bovill JG "Fentanyl and convulsions." Anesth Analg 62 (1983): 858-9
  • "Product Information. Alfenta (alfentanil)." Janssen Pharmaceutica, Titusville, NJ.
  • Smith NT, Benthuysen JL, Bickford RG, Sanford TJ, Blasco T, Duke PC, Head N, Dec-Silver H "Seizures during opioid anesthetic induction--are they opioid-induced rigidity?" Anesthesiology 71 (1989): 852-62
  • Goroszeniuk T, Albin M, Jones RM "Generalized grand mal seizure after recovery from uncomplicated fentanyl-etomidate anesthesia." Anesth Analg 65 (1986): 979-81
  • "Product Information. Dolophine (methadone)." Lilly, Eli and Company, Indianapolis, IN.
  • "Product Information. Kadian (morphine)." Zeneca Pharmaceuticals, Wilmington, DE.
  • "Product Information. Stadol (butorphanol)." Allscrips Pharmaceutical Company, Vernon Hills, IL.
  • "Product Information. Levo-Dromoran (levorphanol)." Roche Laboratories, Nutley, NJ.
  • Hagmeyer KO, Mauro LS, Mauro VF "Meperidine-related seizures associated with patient-controlled analgesia pumps." Ann Pharmacother 27 (1993): 29-32
  • "Product Information. Ultiva (remifentanil)." Mylan Institutional (formally Bioniche Pharma USA Inc), Canonsburg, PA.
  • Stone PA, Macintyre PE, Jarvis DA "Norpethidine toxicity and patient controlled analgesia." Br J Anaesth 71 (1993): 738-40
  • Safwat AM, Daniel D "Grand mal seizure after fentanyl administration." Anesthesiology 59 (1983): 78
  • "Product Information. Vicoprofen (hydrocodone-ibuprofen)." Knoll Pharmaceutical Company, Whippany, NJ.
  • "Product Information. Dilaudid (hydromorphone)." Knoll Pharmaceutical Company, Whippany, NJ.
  • Hoien AO "Another case of grand mal seizure after fentanyl administration." Anesthesiology 60 (1984): 387-8
  • Mauro VF, Bonfiglio MF, Spunt AL "Meperidine-induced seizure in a patient without renal dysfunction or sickle cell anemia." Clin Pharm 5 (1986): 837-9
  • "Product Information. Numorphan (oxymorphone)" Endo Laboratories LLC, Chadds Ford, PA.
  • Reutens DC, Stewart-Wynne EG "Norpethidine induced myoclonus in a patient with renal failure." J Neurol Neurosurg Psychiatry 52 (1989): 1450-1
  • "Product Information. Sublimaze (fentanyl)." Janssen Pharmaceutica, Titusville, NJ.
  • "Product Information. Orlaam (levomethadyl acetate)" Roxanne Laboratories Inc, Columbus, OH.
  • "Product Information. Fentanyl Oralet (fentanyl)." Abbott Pharmaceutical, Abbott Park, IL.
  • Kaiko RF, Foley KM, Grabinski PY, et al "Central nervous system excitatory effects of meperidine in cancer patients." Ann Neurol 13 (1983): 180-5
  • "Product Information. Roxanol (morphine)." Roxane Laboratories Inc, Columbus, OH.
  • Goetting MG, Thirman MJ "Neurotoxicity of meperidine." Ann Emerg Med 14 (1985): 1007-9
  • "Product Information. OxyContin (oxycodone)." Purdue Frederick Company, Norwalk, CT.
  • Sjogren P, Dragsted L, Christensen CB "Myoclonic spasms during treatment with high doses of intravenous morphine in renal failure." Acta Anaesthesiol Scand 37 (1993): 780-2
  • Benthuysen JL, Stanley TH "Concerning the possible nature of reported fentanyl seizures." Anesthesiology 62 (1985): 205
  • "Product Information. Calcidrine (codeine)." Abbott Pharmaceutical, Abbott Park, IL.
  • "Product Information. Duragesic Transdermal System (fentanyl)." Janssen Pharmaceutica, Titusville, NJ.
  • "Product Information. Stadol (butorphanol nasal)." Bristol-Myers Squibb, Princeton, NJ.
  • "Product Information. Buprenex (buprenorphine)." Reckitt and Colman Pharmaceutical, Richmond, VA.
  • Babul N, Darke AC "Putative role of hydromorphone metabolites in myoclonus." Pain 51 (1992): 260-1
  • "Product Information. Opium Tincture (opium)" Lilly, Eli and Company, Indianapolis, IN.
  • "Product Information. Nubain (nalbuphine)." Endo Laboratories, Texarkana, TX.
  • "Product Information. MS Contin (morphine)." Purdue Frederick Company, Norwalk, CT.
  • "Product Information. Talwin NX (pentazocine)." Sanofi Winthrop Pharmaceuticals, New York, NY.
  • "Product Information. Demerol (meperidine)." Sanofi Winthrop Pharmaceuticals, New York, NY.
  • "Product Information. Sufenta (sufentanil)." Janssen Pharmaceutica, Titusville, NJ.
  • Rao TL, Mummaneni N, El-Etr AA "Convulsions: an unusual response to intravenous fentanyl administration." Anesth Analg 61 (1982): 1020-1
Meperidine and Promethazine Capsules

Nome genérico: meperidine / promethazine

Marca comercial:

Sinônimos: Meperidine and Promethazine

Meperidine and Promethazine Capsules <> Distúrbios convulsivos
Relevância: 23.07.2019 Revisor: Shkutko P.M., M.D., in

Na verificação da interação, conforme informações das fontes confiáveis como Drugs.com, Rxlist.com, Webmd.com, Medscape.com, foram identificadas as contra-indicações ou efeitos colaterais que podem prejudicar a saúde ou aumentar efeito negativo ao consumir o medicamento com esta doença concomitante.

Consumidor:

As fenotiazinas podem baixar o limiar convulsivo e induzir convulsões, particularmente quando as doses são elevadas ou aumentou rapidamente e durante o início da terapia. Das fenotiazinas utilizado no tratamento da psicose, clorpromazina parece ter o maior epileptogenic potencial, enquanto fluphenazine e thioridazine que têm menos. A terapia com fenotiazinas deve ser administrado com cautela em pacientes com história de convulsões ou outros fatores de predisposição para convulsões como EEG anormal, preexistente CNS patologia ou traumatismo na cabeça. Adequada terapia anticonvulsivante deve ser mantida durante a administração de fenotiazinas.

Referências
  • DiPiro JT, Talbert RL, Yee GC, Matzke GR, Wells BG, Posey LM "Pharmacotherapy: A Pathophysiologic Approach 4th" Stamford, CT: Appleton & Lange (1999):
  • "Product Information. Tacaryl (methdilazine)." Westwood Squibb Pharmaceutical Corporation, Buffalo, NY.
  • "Product Information. Serentil (mesoridazine)" Boehringer-Ingelheim, Ridgefield, CT.
  • "Product Information. Vesprin (triflupromazine)" Bristol-Myers Squibb, Princeton, NJ.
  • "Product Information. Mellaril (thioridazine)." Sandoz Pharmaceuticals Corporation, East Hanover, NJ.
  • "Product Information. Moban (molindone)." Gate Pharmaceuticals, Sellersville, PA.
  • "Product Information. Stelazine (trifluoperazine)" SmithKline Beecham, Philadelphia, PA.
  • "Product Information. Phenergan (promethazine)." Wyeth-Ayerst Laboratories, Philadelphia, PA.
  • "Product Information. Sparine (promazine)." Wyeth-Ayerst Laboratories, Philadelphia, PA.
  • "Product Information. Prolixin (fluphenazine)." Bristol-Myers Squibb, Princeton, NJ.
  • "Product Information. Torecan (thiethylperazine)" Roxane Laboratories Inc, Columbus, OH.
  • "Product Information. Compazine (prochlorperazine)." SmithKline Beecham, Philadelphia, PA.
  • Markowitz J, Brown R "Seizures with neuroleptics and antidepressants." Gen Hosp Psychiatry 9 (1987): 135-41
  • "Product Information. Trilafon (perphenazine)" Schering Corporation, Kenilworth, NJ.
  • "Product Information. Temaril (trimeprazine)" Allergan Inc, Irvine, CA.
  • Waterhouse RG "Epileptiform convulsions in children following premedication with Pamergan SP100." Br J Anaesth 39 (1967): 268-70
  • "Product Information. Thorazine (chlorpromazine)." SmithKline Beecham, Philadelphia, PA.
  • "Product Information. Orap Tablets (pimozide)." Gate Pharmaceuticals, Sellersville, PA.
Meperidine and Promethazine Capsules

Nome genérico: meperidine / promethazine

Marca comercial:

Sinônimos: Meperidine and Promethazine

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